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1)  Colon-targeted preparation
结肠靶向制剂
2)  oral colon target preparations
口服结肠靶向制剂
3)  colon targeting
结肠靶向
1.
Preparation of Kangfuxin colon targeting micro-pellets;
康复新结肠靶向微丸的制备工艺
2.
In vivo/in vitro evaluation of Kangfuxin colon targeting capsules;
康复新结肠靶向胶囊的体内外评价
3.
Conclusions: This research provided a way for traditional Chinese drug preparation of colon targeting.
目的 :考察中药制备结肠靶向给药的可能。
4)  colon specific
结肠靶向
1.
In this article , a review of research in the colon specific drug delivery based on azo polymers in which azo groups are located in the main chain, cross links, or in branches, is given.
在人体消化道中 ,偶氮键仅能被结肠厌氧菌代谢的偶氮还原酶还原而断裂 ,偶氮聚合物可作为潜在的高定位性的结肠靶向药物缓释载体。
2.
Azo polymers may be expected as colon specific drug delivery systems because azo bonds in polymers can be reduced by azoreductase generated by colonic bacteria.
偶氮聚合物中的偶氮键可被结肠菌丛产生的偶氮还原酶催化还原 ,可用作高定位性的结肠靶向给药药物载体。
5)  colon-specific
结肠靶向
1.
Polysaccharides are used as colon-specific drug delivery carriers because they can be degraded by enzymes produced by colon bacteria.
多糖能被结肠内的菌群降解,而被用作结肠靶向给药的载体。
2.
The aim of this work was to investigate guar gum/ethylcellulose mix coated pellets for potential colon-specific drug delivery.
体外研究瓜尔胶/乙基纤维素混合包衣小丸的结肠靶向性。
3.
slected different properties chemical elements as model drugs,and in view of above problems,studied systematically by free film and membrane controlled preparation according to the requirement of colon-specific.
针对当前膜控材料在中药结肠靶向给药系统中应用的相关性质、影响因素及其与药物匹配性认识不足的问题,本论文以pH敏感型和酶触发型材料为研究对象,以不同性质的化学组分为模型药物,根据结肠递药的要求,从游离膜和膜控制剂两种形式对上述问题进行系统研究,并分析两种形式下研究结果的相关性,揭示各膜控材料用于结肠靶向给药的相关性质及其影响因素,明确其在中药结肠靶向制剂中的适宜性,为中药膜控型结肠靶向制剂的设计、制备提供科学依据。
6)  colon-targeted
结肠靶向
1.
Verification of colon-targeted release of Changankang Pellets;
肠安康微丸结肠靶向验证实验
补充资料:靶制剂
分子式:
CAS号:

性质:具有靶向性的药物制剂称为靶制剂。可为两种类型:(1)药物本身具有特殊性,对机体靶组织有定向亲和作用;(2)借助于载体使药物具靶向性,到达特定的部位起治疗作用。靶制剂由于对组织有亲和性与选择性,其可减少药物使用过量,降低毒性,减轻不良反应,延长药物作用时间,提高治疗效果。

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