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1)  histone deacetylase inhibitor
组蛋白脱乙酰基酶抑制剂
2)  Histone Deacetylase Inhibitor
组蛋白脱乙酰酶抑制剂
3)  5-aza-cytidine
组蛋白脱乙酰化酶抑制剂
1.
DNA methyltransferase (DNMT) inhibitor, 5-aza-cytidine (5-aza-C), was widely studied because DNA hypomethylation induced the re-activation of tumor suppressor genes that were silenced by methylation-mediated mechanisms, could inhibit proliferation and induce differentiation of tumor.
组蛋白脱乙酰化酶抑制剂苯丁酸钠(sodium phenylbutyrate,SPB)通过对组蛋白去乙酰化酶(histone seacetylase,HDAC)的抑制而达到对肿瘤细胞的生长抑制、诱导分化及诱导凋亡的作用。
4)  histone deacetylase inhibitors
组蛋白去乙酰酶抑制剂
1.
Progress in the research of histone deacetylase inhibitors;
组蛋白去乙酰酶抑制剂的研究进展
5)  histone deacetylase(HDAC) inhibitor
组蛋白乙酰酶抑制剂
6)  histone deacetylase inhibitors
组蛋白去乙酰化酶抑制剂
1.
Mechanism of histone deacetylase inhibitors for treatment of hematological cancer and their clinical research;
组蛋白去乙酰化酶抑制剂治疗血液系统肿瘤的作用机制及临床应用
2.
Molecular mechanism of p21~(WAF1/CIP1) expression induced by histone deacetylase inhibitors in HeLa cell line;
组蛋白去乙酰化酶抑制剂诱导H eLa细胞p21~(WAF1/CIP1)表达的分子机制研究
3.
Mechanism of regulating multidrug resistances by histone deacetylase inhibitors in tumor cells;
组蛋白去乙酰化酶抑制剂调节肿瘤细胞多药耐药性的机制
补充资料:多巴脱羧酶抑制剂
分子式:
CAS号:

性质:能够抑制多巴脱羧酶活性的一类化学物质,如在曲霉和链霉菌发酵液中发现的一类异黄酮,能够非特异性地抑制多巴脱羧酶活性,对自发性高血压的大鼠有降压作用,活性大小与α-甲基多巴胺相当。

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